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p38-alfa MAPK-IN-1

T12347
TargetMol Chemicals
CAS Number443913-15-3
Product group Chemicals
Molecular Weight477.6
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Packing Size
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Overview

  • Supplier
    TargetMol Chemicals
  • Product Name
    p38-alfa MAPK-IN-1
  • Delivery Days Customer
    9
  • CAS Number
    443913-15-3
  • Category Supplier
    Chemical
  • Chemical Name
    p38-alfa MAPK-IN-1
  • Molecular Formula
    C27H35N5O3
  • Molecular Weight
    477.6
  • Scientific Description
    p38-alfa MAPK-IN-1 is a MAPK14 (p38-alfa) inhibitor with IC50 of 2300 nM and 5500 nM in EFC displacement assay and HTRF assay,respectively.
  • Shelf life instruction
    3 years
  • SMILES
    N(C(NC1=CC=C(OCCN2CCOCC2)C=C1)=O)C=3N(N=C(C(C)(C)C)C3)C4=CC=C(C)C=C4
  • Storage Instruction
    -20°
  • UNSPSC
    12352200

References

  • Kluter S, et al. Displacement assay for the detection of stabilizers of inactive kinase conformations. J Med Chem. 2010 Jan 14;53(1):357-67.